郑月钦
学术博士生导师
职称:教授
***
学院:多靶标天然药物全国重点实验室
yzheng@cpu.edu.cn
招生学科:药物化学,药学-药物合成与工艺优化
https://www.x-mol.com/groups/ZhengLab
个人简介

郑月钦,博士,教授,博士生导师,国家青年特聘专家(中组部),江苏特聘教授

中国药科大学孟目的学院副院长,天然药物活性组分与药效国家重点实验室课题组组长                                                                                                   

出生日期:198812

电话: (86) 15851854569

邮件yueqinzheng@hotmail.com;  yzheng@cpu.edu.cn

课题组网站:https://www.x-mol.com/groups/ZhengLab/publications

                        

教育和科研经历

中国药科大学                                                                                                          教授         2020-now

 

哈佛医学院,麻省理工学院                                                                         博士后研究员   2018- 2020                                                              

合作导师: Daniel Kohane 教授(Harvard);Robert S. Langer 教授(MIT

 

美国佐治亚州立大学                                                                                            博士生        2012-2017

合作导师王炳和教授

 

中国科学技术大学                                                                                                    学士         2007-2011

指导老师:汪志勇教授

 

荣誉与奖项

2021   江苏省特聘教授

2020    国家重大人才工程A 青年项目

2018    中国优秀自费留学生奖学金

2017    佐治亚州立大学研究生学生金奖

 

主持项目

国家重大人才工程A类项目(2020-2023);

国家自然科学基金项目 (2021-2024);

江苏省自然科学基金项目 (2021-2024);

海外高层次人才引进项目  (2020-2025);

国家自然科学基金项目 (2024-2027);

国家自然科学基金项目 (2026-2029);


近期代表性论文

1. Jianru Liu+,Yuanan Wang+, Qiwei Zhou,Wen Peng,Peiyuan Li,Chao Ban,Yangyin Xue,Yan Liang,Zhongbo Wang,Hao Hao,Yanzhao Chen,Weiwei Guo*,Yueqin Zheng*, Precursors of Carboximidates Deriving from Thioamide-Trimethyl-Lock System: A General Method for Designing Stable Cascade Acid-Sensitive Prodrugs. J. Am. Chem. Soc. 2025,  https://doi.org/10.1021/jacs.5c03565.


2. Xiaowei Xu,? Yuanan Wang,? Yangfei Shi, Xin Wang, Xidan Tong, Yanzhao Chen, Yan Zhao, 4 Jiaxuan Chen, Weiwei Guo, and Yueqin Zheng*,Development of Cyclooctyne-Nitrone Based Click Release Chemistry for Bioorthogonal Prodrug Activation both In Vitro and In Vivo, J. Am. Chem. Soc. 2025,https://doi.org/10.1021/jacs.5c08152.


3. Wen Peng, Lixiao Qin, Tianci Wang, Yangqian Sun, Zhen Li, David J. Lefer, Cheng Luo, Fei Ye, Binghe Wang*, Weiwei Guo* ,Yueqin Zheng*,  A Highly Atom-Efficient Prodrug Approach to Generate Synergy between H2S and Nonsteroidal Anti-inflammatory Drugs and Improve Safety. J. Med. Chem. 2024, 67, 19, 17350–17362. https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c01254.

4. Xidan Tong, Jiaxuan Chen, Maolin Wang, Jianru Liu, Jing Li, Xin Wang, Yifei Zuo, Xiaowei Xu, Yichen Wang, Binghe Wang*, Weiwei Guo*, Yueqin Zheng*, Development of a Bioorthogonal Click-to-Release Reaction for Hydrogen Polysulfide (H2Sn) Detection. Anal. Chem. 2024, 96, 39, 15631–15639.  https://pubs.acs.org/doi/10.1021/acs.analchem.4c02677.

5. Wen Peng, Jianru Liu, Zhen Li, Yuanan Wang, Yangqian Sun, Yanzhao Chen, David J. Lefer*, Weiwei Guo*, Yueqin Zheng*,A Bifunctional Sulfide Donor Approach for Ischemic Stroke: Leveraging Butylphthalide as a Carrier for Sulfide Prodrug, J. Med. Chem. 2024, 67, 22, 20695–20707https://doi.org/10.1021/acs.jmedchem.4c02454

6. Jing Li+, Mingxin Cheng+, Hongbo Zhang, Yichen Wang, Weiwei Guo*, and Yueqin Zheng*,A Tetrazine Amplification System for Visual Detection of Trace Analytes via Click-Release Reactions. Angewandte Chemie International Edition. 2024. https://doi.org/10.1002/anie.202414246




 

个人经历
科研项目
科研专利
发表论文
获奖成果
教材专著

研究方向

课题组研究聚焦于新型化学生物学在疾病的诊断和治疗方向的研究包括 :设计硫化氢前药用于治疗心脑血管疾病的研究;开发新生物正交化学用于疾病的诊断和药物的开发;开发长效选择性感觉神经阻滞的局部麻药等